Bayyanar / launi: fari mai ƙarfi
● Tarihi matsa lamba: 0.00232MMHG a 25 ° C
Point ● Melting Points: 285-286 ° C (Dec.) (Lit.)
Indeve Index: 1.7990 (kimanta)
● Poust Point: 288.5 ° C a 760 mmhg
● Pka: 10.61 ± 0.50 (annabta)
● FASTT FASHT: 128.3 ° C
● PISA: 98.05000
● Tecity: 1.84 g / cm3
● Laja: 0.50900
● Storge Temp.:desicccccccate a + 4 ° C
● Mai hankali .::::::::::::::::5
● Sulurility.:DMO (dan kadan), methanol (dan kadan)
● Picogram (s):Xi
Lambobin Hadiki: Xi
● Bayani: 36/37/38
Bayanin Tsaro: 22-24 / 25-36-26
Bayanin: 2,4-Diamoxypypedine 2-Hydroxypypedine (Dahp) ne mai zaɓa, takamaiman inhih na GTP Cyclohydrase i, ragin karuwa mataki don de novo pterin synthesis. A cikin sel, IC50 don hana bh4 biosynthesis kusan 0.3 mm. Ana iya amfani da Dahp don toshe cikin yadda ake samarwa a cikin nau'ikan tantanin halitta da yawa.
● Amfani da: 2,4-Diamoxypypedine (Dahp) mai zabi ne, takamaiman inhih na GTP Cyclohydrase I, da ragin iyakance mataki don de novo pterin synthesis. A cikin sel, IC50 don hana bh4 biosynthesis kusan 0.3 mm. Ana iya amfani da Dahp don toshe cikin yadda ya kamata babu wani samarwa a cikin nau'ikan tantanin halitta da yawa. [Carrosine, da Trypalo-6-hydroxypyfydine, Tydroxypyfydine, Tydroxypypedine wannan a cikin tsarin kwayar halitta.
2,4-Diramo-6-Hydroxypypedine shine fili mai guba tare da tsarin ƙwayar ƙwayar C4h6No. Ana amfani dashi azaman tsaka-tsaki a cikin tsarin mahadi daban-daban, gami da magunguna masu zobe guda biyu (NH2) da rukunin Hydroxyl guda biyu (OH) Hyedroxyl rukuni (oh) a haɗe zuwa carbon carbon na carbon daban-daban. Wannan tsarin ya sa ya zama toshewar ginin da ke tattare da sernan kwayoyin halitta.2,4-Dimano-6-hydroxypypyens daban-daban, gami da dauki cyanamide tare da urea. Tana da aikace-aikace da yawa a masana'antar harhada magunguna, musamman a cikin magungunan maganin, musamman a cikin magungunan maganin, ƙwayoyin cuta, 2,4-Diamoroxype-6-hyyroxypypyine ne mai mahimmanci a cikin aikace-aikacen sunadarai da magunguna da magunguna.
2,4-Diramo-6-Hydroxypypedine shine fili mai guba tare da tsarin ƙwayar ƙwayar C4h6No. Yana da kwali na kwayoyin halitta na dangin PyrimIDine ne. Gobalin yana da tsarin zobe na pyrimine, ƙungiyoyi biyu (NH2) an haɗa su a matsayi na 2 da 4-matsayi (oh) an haɗa su a matsayi na 6. Za'a iya bayyana tsarin sunadarai kamar: ammoniya | | H - C - C - C - N - C - C - NH2 | | Oh 2,4-Diamero-6-Hydroxypypa'idine yana da aikace-aikace iri-aikace daban-daban a cikin masana'antar harhada magunguna. Yana da mahimmanci matsakaici a cikin tsarin magunguna, ciki har da antitistorist da magunguna masu maganin antitistor. Hakanan ana amfani dashi don samar da analogs da yawa da aka yi amfani da su a cikin binciken magunguna.
Baya ga aikace-aikacen aikace-aikacen magunguna, 2,4-Diamo-6-hydroxypypidine shima ana amfani dashi azaman sinadaran a cikin agrochemicalicals. Sadarwar take a cikin tsarin da ke tattare da kayan gargajiya da fungicides. Yana da matukar muhimmanci a bi ingantaccen tsarin aminci lokacin amfani da 2,4-dimano-6-hydroxypypyine. Tunda an rarraba shi a matsayin m, yakamata a kula da shi da kuma isasshen kayan kariya na mutum ya kamata a sawa don guje wa kai tsaye.
A taƙaice, 2,4-Diamino-6-hydroxypypyine shine fili na kwayoyin tare da aikace-aikace a cikin fannoni na aikin gona da gonar gona. Tsarin sunadarai yana sa yana da amfani azaman tsaka-tsaki a cikin tsarin magunguna da tsiro masu rikitarwa.